Thomas Jefferson University

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Peiper, Stephen
One or more keywords matched the following items that are connected to Peiper, Stephen
Item TypeName
Concept Oligopeptides
Academic Article A point mutation that confers constitutive activity to CXCR4 reveals that T140 is an inverse agonist and that AMD3100 and ALX40-4C are weak partial agonists.
Academic Article Molecular-size reduction of a potent CXCR4-chemokine antagonist using orthogonal combination of conformation- and sequence-based libraries.
Academic Article Lipid bilayer simulations of CXCR4 with inverse agonists and weak partial agonists.
Academic Article Synthesis of potent CXCR4 inhibitors possessing low cytotoxicity and improved biostability based on T140 derivatives.
Academic Article Enhancement of the T140-based pharmacophores leads to the development of more potent and bio-stable CXCR4 antagonists.
Academic Article Topochemical exploration of potent compounds using retro-enantiomer libraries of cyclic pentapeptides.
Academic Article Identification of novel low molecular weight CXCR4 antagonists by structural tuning of cyclic tetrapeptide scaffolds.
Academic Article Kisspeptin-10-induced signaling of GPR54 negatively regulates chemotactic responses mediated by CXCR4: a potential mechanism for the metastasis suppressor activity of kisspeptins.
Academic Article Development of a linear type of low molecular weight CXCR4 antagonists based on T140 analogs.
Academic Article SAR and QSAR studies on the N-terminally acylated pentapeptide agonists for GPR54.
Academic Article KiSS1 metastasis suppressor gene product induces suppression of tyrosine kinase receptor signaling to Akt, tumor necrosis factor family ligand expression, and apoptosis.
Academic Article Activation of Rho and Rho-associated kinase by GPR54 and KiSS1 metastasis suppressor gene product induces changes of cell morphology and contributes to apoptosis.
Academic Article Expression of CXCR4, a G-protein-coupled receptor for CXCL12 in yeast identification of new-generation inverse agonists.
Academic Article Structure-activity relationship study on artificial CXCR4 ligands possessing the cyclic pentapeptide scaffold: the exploration of amino acid residues of pentapeptides by substitutions of several aromatic amino acids.
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  • Oligopeptides